Discovery of a targeted covalent CDK14 inhibitor with a TAIRE kinase-biased selectivity profile Aug. 30, 2019 No Comments
SU-011 improves glycemic control in vivo without the risk of hypoglycemia and weight gain Aug. 20, 2019 No Comments
DS-39201083 is a new derivative of conolidine with superior analgesic activity Aug. 14, 2019 No Comments
TR-FRET-based screening identifies novel CBP bromodomain inhibitor with therapeutic potential Aug. 13, 2019 No Comments
Novel M4 positive allosteric modulator with improved physicochemical properties and favorable PK Aug. 9, 2019 No Comments
Small molecule WX2-43 targets PRMT5-KLF4 for triple-negative breast cancer treatment Aug. 6, 2019 No Comments
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